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Amodiaquine dihydrochloride

Glpbio
Catalog No:GC60579-10mM (in 1mL DMSO) CAS No.:69-44-3 MDLNo:C20H24Cl3N3O Brand:Glpbio purity: 特性: Purpose:Amodiaquinedihydrochloride(Amodiaquindihydrochloride)是一种4-氨基喹啉类抗疟剂,是一种有效的具有口服活性的组胺N-甲基转移酶(histamineN-methyltransferase)抑制剂,Ki值为18.6nM。Amodiaquinedihydrochloride也是一种Nurr1激动剂,可特异性结合Nurr1的配体结合域,EC50为~20μM。抗炎作用。DMSO: 125 mg/mL (291.52 mM; Need ultrasonic)
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